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U-47700 is an opioid analgesic that was first developed by Upjohn about 40 years ago. It is derived from the related opioid, AH-7921. Despite its importance in the development of this class of opioid chemicals, U-47700 itself has never been officially tested on humans or animals.
Pharmacology:
U-47700 is highly selective for -opioid receptors and is believed to be about 7 to 8 times more potent than morphine per dose. It is considered a strong kappa agonist, so it should not cause significant levels of dysphoria or other side effects.
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